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A2A receptor antagonist 1

CAS No. 443103-97-7

A2A receptor antagonist 1( CPI-444 analog )

Catalog No. M28146 CAS No. 443103-97-7

A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 87 Get Quote
10MG 140 Get Quote
25MG 293 Get Quote
50MG 447 Get Quote
100MG 664 Get Quote
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Biological Information

  • Product Name
    A2A receptor antagonist 1
  • Note
    Research use only, not for human use.
  • Brief Description
    A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
  • Description
    A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.(In Vitro):A2A receptor anyagonist 1 is a potent adenosine A2A receptor antagonist, selective over the A1 receptor and demonstrate its binding activity with Ki values of 4 and 264 nM, respectively.
  • In Vitro
    A2A receptor antagonist 1 (CPI-444 analog)?is a potent adenosine A2A receptor antagonist, selective over the A1 receptor and demonstrates its binding activity with Ki values of 4 and 264 nM, respectively.
  • In Vivo
    ——
  • Synonyms
    CPI-444 analog
  • Pathway
    Apoptosis
  • Target
    Adenosine Receptor
  • Recptor
    MAGL
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    443103-97-7
  • Formula Weight
    309.3
  • Molecular Formula
    C16H12FN5O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 25 mg/mL (80.83 mM)
  • SMILES
    Nc1nc(-c2ccco2)c2cnn(Cc3ccccc3F)c2n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Aaltonen N, et al. Piperazine and piperidine triazole ureas as ultrapotent and highly selective inhibitors of monoacylglycerol lipase. Chem Biol. 2013 Mar 21;20(3):379-90.
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