Cart
sales@molnova.com
Home - Products - Apoptosis - Adenosine Receptor - A2A receptor antagonist 1

A2A receptor antagonist 1

CAS No. 443103-97-7

A2A receptor antagonist 1( CPI-444 analog )

Catalog No. M28146 CAS No. 443103-97-7

A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 87 Get Quote
10MG 140 Get Quote
25MG 293 Get Quote
50MG 447 Get Quote
100MG 664 Get Quote
500MG 1395 Get Quote
1G Get Quote Get Quote
Get Quotation Bulk Inquiry Add to Cart

Biological Information

  • Product Name
    A2A receptor antagonist 1
  • Note
    Research use only, not for human use.
  • Brief Description
    A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
  • Description
    A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.(In Vitro):A2A receptor anyagonist 1 is a potent adenosine A2A receptor antagonist, selective over the A1 receptor and demonstrate its binding activity with Ki values of 4 and 264 nM, respectively.
  • In Vitro
    A2A receptor antagonist 1 (CPI-444 analog)?is a potent adenosine A2A receptor antagonist, selective over the A1 receptor and demonstrates its binding activity with Ki values of 4 and 264 nM, respectively.
  • In Vivo
    ——
  • Synonyms
    CPI-444 analog
  • Pathway
    Apoptosis
  • Target
    Adenosine Receptor
  • Recptor
    MAGL
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    443103-97-7
  • Formula Weight
    309.3
  • Molecular Formula
    C16H12FN5O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 25 mg/mL (80.83 mM)
  • SMILES
    Nc1nc(-c2ccco2)c2cnn(Cc3ccccc3F)c2n1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Aaltonen N, et al. Piperazine and piperidine triazole ureas as ultrapotent and highly selective inhibitors of monoacylglycerol lipase. Chem Biol. 2013 Mar 21;20(3):379-90.
Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog
related products

  • CI-947

    An orally active adenosine receptor agonist that can induce acute cardiovascular toxicity and coronary vascular injury in vivo.

  • Derenofylline

    Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM).

  • Tonapofylline

    A potent, selective and orally bioavailable adenosine A1 (A1A) receptor antagonist with Ki of 7 nM.

Sign In Join Free